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Target
Stromal cell-derived factor 1
Ligand
BDBM50572275
Substrate
n/a
Meas. Tech.
ChEMBL_2116663 (CHEMBL4825604)
Kd
3024000±n/a nM
Citation
Sprague, DJ; Getschman, AE; Fenske, TG; Volkman, BF; Smith, BC Trisubstituted 1,3,5-Triazines: The First Ligands of the sY12-Binding Pocket on Chemokine CXCL12. ACS Med Chem Lett 12:1773-1782 (2021) [PubMed] Article
More Info.:
Target
Name:
Stromal cell-derived factor 1
Synonyms:
CXCL12 | Chemokine CXCL12 | SDF1 | SDF1A | SDF1B | SDF1_HUMAN
Type:
Enzyme
Mol. Mass.:
10677.83
Organism:
Human
Description:
P48061
Residue:
93
Sequence:
MNAKVVVVLVLVLTALCLSDGKPVSLSYRCPCRFFESHVARANVKHLKILNTPNCALQIVARLKNNNRQVCIDPKLKWIQEYLEKALNKRFKM