Reaction Details Report a problem with these data
Target
Proteasome subunit alpha type-1
Ligand
BDBM50577116
Substrate
n/a
Meas. Tech.
ChEMBL_2129501 (CHEMBL4838930)
IC50
4356±n/a nM
Citation
More Info.:
Target
Name:
Proteasome subunit alpha type-1
Synonyms:
30 kDa prosomal protein | HC2 | Macropain subunit C2 | Multicatalytic endopeptidase complex subunit C2 | NU | PROS-30 | PROS30 | PSA1_HUMAN | PSC2 | PSMA1 | Proteasome component C2 | Proteasome nu chain
Type:
PROTEIN
Mol. Mass.:
29555.77
Organism:
Homo sapiens (Human)
Description:
ChEMBL_106197
Residue:
263
Sequence:
MFRNQYDNDVTVWSPQGRIHQIEYAMEAVKQGSATVGLKSKTHAVLVALKRAQSELAAHQKKILHVDNHIGISIAGLTADARLLCNFMRQECLDSRFVFDRPLPVSRLVSLIGSKTQIPTQRYGRRPYGVGLLIAGYDDMGPHIFQTCPSANYFDCRAMSIGARSQSARTYLERHMSEFMECNLNELVKHGLRALRETLPAEQDLTTKNVSIGIVGKDLEFTIYDDDDVSPFLEGLEERPQRKAQPAQPADEPAEKADEPMEH