Reaction Details Report a problem with these data
Target
Sigma intracellular receptor 2
Ligand
BDBM50584893
Substrate
n/a
Meas. Tech.
ChEMBL_2160848 (CHEMBL5045598)
Ki
1000±n/a nM
Citation
Wen, Z; Salmaso, V; Jung, YH; Phung, NB; Gopinatth, V; Shah, Q; Patterson, AT; Randle, JCR; Chen, Z; Salvemini, D; Lieberman, DI; Whitehead, GS; Karcz, TP; Cook, DN; Jacobson, KA Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y J Med Chem 65:3434-3459 (2022) [PubMed] Article
More Info.:
Target
Name:
Sigma intracellular receptor 2
Synonyms:
MAC30 | Meningioma-associated protein 30 | S2R | SGMR2_HUMAN | Sigma-2 receptor | Sigma2 receptor | TMEM97 | Transmembrane protein 97
Type:
Protein
Mol. Mass.:
20857.20
Organism:
Homo sapiens (Human)
Description:
Q5BJF2
Residue:
176
Sequence:
MGAPATRRCVEWLLGLYFLSHIPITLFMDLQAVLPRELYPVEFRNLLKWYAKEFKDPLLQEPPAWFKSFLFCELVFQLPFFPIATYAFLKGSCKWIRTPAIIYSVHTMTTLIPILSTFLFEDFSKASGFKGQRPETLHERLTLVSVYAPYLLIPFILLIFMLRSPYYKYEEKRKKK