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Target
Triosephosphate isomerase
Ligand
BDBM50167775
Substrate
n/a
Meas. Tech.
ChEMBL_302548 (CHEMBL828250)
Ki
4500±n/a nM
Citation
Fonvielle, M; Mariano, S; Therisod, M New inhibitors of rabbit muscle triose-phosphate isomerase. Bioorg Med Chem Lett 15:2906-9 (2005) [PubMed] Article
More Info.:
Target
Name:
Triosephosphate isomerase
Synonyms:
TPI1 | TPIS_RABIT
Type:
PROTEIN
Mol. Mass.:
26758.31
Organism:
Rabbit
Description:
ChEMBL_302548
Residue:
249
Sequence:
MAPSRKFFVGGNWKMNGRKKNLGELITTLNAAKVPADTEVVCAPPTAYIDFARQKLDPKIAVAAQNCYKVTNGAFTGEISPGMIKDCGATWVVLGHSERRHVFGESDELIGQKVAHALSEGLGVIACIGEKLDEREAGITEKVVFEQTKVIADNVKDWSKVVLAYEPVWAIGTGKTATPQQAQEVHEKLRGWLKSNVSDAVAQSTRIIYGGSVTGATCKELASQPDVDGFLVGGASLKPEFVDIINAKQ