Reaction Details Report a problem with these data
Target
EEF1AKMT4-ECE2 readthrough transcript protein
Ligand
BDBM50271178
Substrate
n/a
Meas. Tech.
ChEMBL_552748 (CHEMBL965254)
IC50
5830±n/a nM
Citation
Gagnidze, K; Sachchidanand, na; Rozenfeld, R; Mezei, M; Zhou, MM; Devi, LA Homology modeling and site-directed mutagenesis to identify selective inhibitors of endothelin-converting enzyme-2. J Med Chem 51:3378-87 (2008) [PubMed] Article
More Info.:
Target
Name:
EEF1AKMT4-ECE2 readthrough transcript protein
Synonyms:
EEF1AKMT4-ECE2 | EFCE2_HUMAN | Endothelin-converting enzyme 2 | Endothelin-converting enzyme 2 (ECE-2) | Endothelin-converting enzyme 2 (ECE2) | Endothelin-converting enzyme 2 region
Type:
Enzyme
Mol. Mass.:
99745.05
Organism:
Human
Description:
P0DPD8
Residue:
883
Sequence:
MASPGAGRAPPELPERNCGYREVEYWDQRYQGAADSAPYDWFGDFSSFRALLEPELRPEDRILVLGCGNSALSYELFLGGFPNVTSVDYSSVVVAAMQARHAHVPQLRWETMDVRKLDFPSASFDVVLEKGTLDALLAGERDPWTVSSEGVHTVDQVLSEVGFQKGTRQLLGSRTQLELVLAGASLLLAALLLGCLVALGVQYHRDPSHSTCLTEACIRVAGKILESLDRGVSPCEDFYQFSCGGWIRRNPLPDGRSRWNTFNSLWDQNQAILKHLLENTTFNSSSEAEQKTQRFYLSCLQVERIEELGAQPLRDLIEKIGGWNITGPWDQDNFMEVLKAVAGTYRATPFFTVYISADSKSSNSNVIQVDQSGLFLPSRDYYLNRTANEKVLTAYLDYMEELGMLLGGRPTSTREQMQQVLELEIQLANITVPQDQRRDEEKIYHKMSISELQALAPSMDWLEFLSFLLSPLELSDSEPVVVYGMDYLQQVSELINRTEPSILNNYLIWNLVQKTTSSLDRRFESAQEKLLETLYGTKKSCVPRWQTCISNTDDALGFALGSLFVKATFDRQSKEIAEGMISEIRTAFEEALGQLVWMDEKTRQAAKEKADAIYDMIGFPDFILEPKELDDVYDGYEISEDSFFQNMLNLYNFSAKVMADQLRKPPSRDQWSMTPQTVNAYYLPTKNEIVFPAGILQAPFYARNHPKALNFGGIGVVMGHELTHAFDDQGREYDKEGNLRPWWQNESLAAFRNHTACMEEQYNQYQVNGERLNGRQTLGENIADNGGLKAAYNAYKAWLRKHGEEQQLPAVGLTNHQLFFVGFAQVWCSVRTPESSHEGLVTDPHSPARFRVLGTLSNSRDFLRHFGCPVGSPMNPGQLCEVW