Reaction Details Report a problem with these data
Target
Phospholipase A2, membrane associated
Ligand
BDBM50274391
Substrate
n/a
Meas. Tech.
ChEMBL_537135 (CHEMBL989795)
IC50
>1600±n/a nM
Citation
Oslund, RC; Cermak, N; Verlinde, CL; Gelb, MH Simplified YM-26734 inhibitors of secreted phospholipase A2 group IIA. Bioorg Med Chem Lett 18:5415-9 (2008) [PubMed] Article
More Info.:
Target
Name:
Phospholipase A2, membrane associated
Synonyms:
PA2GA_RAT | Phospholipase A2 group IIA | Pla2g2a
Type:
PROTEIN
Mol. Mass.:
16307.95
Organism:
Rat
Description:
ChEMBL_537135
Residue:
146
Sequence:
MKVLLLLAVVIMAFGSIQVQGSLLEFGQMILFKTGKRADVSYGFYGCHCGVGGRGSPKDATDWCCVTHDCCYNRLEKRGCGTKFLTYKFSYRGGQISCSTNQDSCRKQLCQCDKAAAECFARNKKSYSLKYQFYPNKFCKGKTPSC