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Target
Phospholipase A2, membrane associated
Ligand
BDBM50274387
Substrate
n/a
Meas. Tech.
ChEMBL_537135 (CHEMBL989795)
IC50
>1600±n/a nM
Citation
 Oslund, RC; Cermak, N; Verlinde, CL; Gelb, MH Simplified YM-26734 inhibitors of secreted phospholipase A2 group IIA. Bioorg Med Chem Lett 18:5415-9 (2008) [PubMed]  Article 
Target
Name:
Phospholipase A2, membrane associated
Synonyms:
PA2GA_RAT | Phospholipase A2 group IIA | Pla2g2a
Type:
PROTEIN
Mol. Mass.:
16307.95
Organism:
Rat
Description:
ChEMBL_537135
Residue:
146
Sequence:
MKVLLLLAVVIMAFGSIQVQGSLLEFGQMILFKTGKRADVSYGFYGCHCGVGGRGSPKDATDWCCVTHDCCYNRLEKRGCGTKFLTYKFSYRGGQISCSTNQDSCRKQLCQCDKAAAECFARNKKSYSLKYQFYPNKFCKGKTPSC
  
Inhibitor
Name:
BDBM50274387
Synonyms:
1-(3-Acetyl-2,4,6-trihydroxy-5-methyl-phenyl)-ethanone | CHEMBL455273
Type:
Small organic molecule
Emp. Form.:
C11H12O5
Mol. Mass.:
224.21
SMILES:
CC(=O)c1c(O)c(C)c(O)c(C(C)=O)c1O
Structure:
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