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Target
Carboxypeptidase A1
Ligand
BDBM50289561
Substrate
n/a
Meas. Tech.
ChEBML_45612
IC50
29000±n/a nM
Citation
 Lanthier, CM; Parniak, MA; Dmitrienko, GI Inhibition of carboxypeptidase a by N-(4-t-Butylbenzoyl)-2-hydroxy-1-naphthaldehyde hydrazone Bioorg Med Chem Lett 7:1557-1562 (1997)    Article 
Target
Name:
Carboxypeptidase A1
Synonyms:
CBPA1_BOVIN | CPA | CPA1 | Carboxypeptidase A | Carboxypeptidase A (CPA) | Carboxypeptidase A1 precursor
Type:
Enzyme
Mol. Mass.:
47073.90
Organism:
Bovine
Description:
From Sigma-Aldrich Co.
Residue:
419
Sequence:
MQGLLILSVLLGAALGKEDFVGHQVLRITAADEAEVQTVKELEDLEHLQLDFWRGPGQPGSPIDVRVPFPSLQAVKVFLEAHGIRYRIMIEDVQSLLDEEQEQMFASQSRARSTNTFNYATYHTLDEIYDFMDLLVAEHPQLVSKLQIGRSYEGRPIYVLKFSTGGSNRPAIWIDLGIHSREWITQATGVWFAKKFTEDYGQDPSFTAILDSMDIFLEIVTNPDGFAFTHSQNRLWRKTRSVTSSSLCVGVDANRNWDAGFGKAGASSSPCSETYHGKYANSEVEVKSIVDFVKDHGNFKAFLSIHSYSQLLLYPYGYTTQSIPDKTELNQVAKSAVEALKSLYGTSYKYGSIITTIYQASGGSIDWSYNQGIKYSFTFELRDTGRYGFLLPASQIIPTAQETWLGVLTIMEHTLNNLY
  
Inhibitor
Name:
BDBM50289561
Synonyms:
4-tert-Butyl-benzoic acid [1-(2-hydroxy-naphthalen-1-yl)-meth-(E)-ylidene]-hydrazide | CHEMBL41643
Type:
Small organic molecule
Emp. Form.:
C22H22N2O2
Mol. Mass.:
346.4223
SMILES:
CC(C)(C)c1ccc(cc1)C(=O)N\N=C\c1c(O)ccc2ccccc12
Structure:
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