Reaction Details Report a problem with these data
Target
Cytosol aminopeptidase [33-68,L62W]
Ligand
BDBM50157555
Substrate
n/a
Meas. Tech.
ChEMBL_546423 (CHEMBL1025822)
IC50
35100±n/a nM
Citation
 Parellada, J; Guinea, M Flavonoid Inhibitors of Trypsin and Leucine Aminopeptidase: A Proposed Mathematical Model for IC50 Estimation J Nat Prod 58:823-829 (1995) [PubMed]  Article 
Target
Name:
Cytosol aminopeptidase [33-68,L62W]
Synonyms:
AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:
Enzyme
Mol. Mass.:
4015.44
Organism:
Sus scrofa (Pig)
Description:
P28839[33-68,L62W]
Residue:
36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
  
Inhibitor
Name:
BDBM50157555
Synonyms:
2-(3,4-dihydroxyphenyl)-4H-chromen-4-one | 3',4'-dihydroxy flavone | 3',4'-dihydroxyflavone | CHEMBL222556
Type:
Small organic molecule
Emp. Form.:
C15H10O4
Mol. Mass.:
254.2375
SMILES:
Oc1ccc(cc1O)-c1cc(=O)c2ccccc2o1
Structure:
Search PDB for entries with ligand similarity: