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Target
Uncharacterized serine/threonine-protein kinase SBK3
Ligand
BDBM50355500
Substrate
n/a
Meas. Tech.
ChEMBL_774227 (CHEMBL1908444)
Kd
>10000±n/a nM
Citation
Davis, MI; Hunt, JP; Herrgard, S; Ciceri, P; Wodicka, LM; Pallares, G; Hocker, M; Treiber, DK; Zarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol 29:1046-51 (2011) [PubMed] Article
More Info.:
Target
Name:
Uncharacterized serine/threonine-protein kinase SBK3
Synonyms:
Putative uncharacterized serine/threonine-protein kinase SgK110 | SBK3 | SBK3_HUMAN | SGK110
Type:
PROTEIN
Mol. Mass.:
38472.62
Organism:
Human
Description:
ChEMBL_774227
Residue:
359
Sequence:
MERRASETPEDGDPEEDTATALQRLVELTTSRVTPVRSLRDQYHLIRKLGSGSYGRVLLAQPHQGGPAVALKLLRRDLVLRSTFLREFCVGRCVSAHPGLLQTLAGPLQTPRYFAFAQEYAPCGDLSGMLQERGLPELLVKRVVAQLAGALDFLHSRGLVHADVKPDNVLVFDPVCSRVALGDLGLTRPEGSPTPAPPVPLPTAPPELCLLLPPDTLPLRPAVDSWGLGVLLFCAATACFPWDVALAPNPEFEAFAGWVTTKPQPPQPPPPWDQFAPPALALLQGLLDLDPETRSPPLAVLDFLGDDWGLQGNREGPGVLGSAVSYEDREEGGSSLEEWTDEGDDSKSGGRTGTDGGAP