Reaction Details Report a problem with these data
Target
Gamma-aminobutyric acid receptor subunit rho-2
Ligand
BDBM50087269
Substrate
n/a
Meas. Tech.
ChEMBL_68705 (CHEMBL682636)
EC50
17500±n/a nM
Citation
Chebib, M; Johnston, GA GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology. J Med Chem 43:1427-47 (2000) [PubMed] Article
More Info.:
Target
Name:
Gamma-aminobutyric acid receptor subunit rho-2
Synonyms:
GABA receptor rho-2 subunit | GABA(A) receptor subunit rho-2 | GABA(C) receptor | GABA-C receptor | GABRR2 | GBRR2_HUMAN | Gamma-aminobutyric acid receptor subunit rho-2
Type:
PROTEIN
Mol. Mass.:
54168.90
Organism:
Human
Description:
ChEMBL_68702
Residue:
465
Sequence:
MPYFTRLILFLFCLMVLVESRKPKRKRWTGQVEMPKPSHLYKKNLDVTKIRKGKPQQLLRVDEHDFSMRPAFGGPAIPVGVDVQVESLDSISEVDMDFTMTLYLRHYWKDERLAFSSASNKSMTFDGRLVKKIWVPDVFFVHSKRSFTHDTTTDNIMLRVFPDGHVLYSMRITVTAMCNMDFSHFPLDSQTCSLELESYAYTDEDLMLYWKNGDESLKTDEKISLSQFLIQKFHTTSRLAFYSSTGWYNRLYINFTLRRHIFFFLLQTYFPATLMVMLSWVSFWIDRRAVPARVSLGITTVLTMTTIITGVNASMPRVSYVKAVDIYLWVSFVFVFLSVLEYAAVNYLTTVQERKERKLREKFPCMCGMLHSKTMMLDGSYSESEANSLAGYPRSHILTEEERQDKIVVHLGLSGEANAARKKGLLKGQTGFRIFQNTHAIDKYSRLIFPASYIFFNLIYWSVFS