Reaction Details
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Target
Tyrosine-protein kinase Blk
Ligand
BDBM50379186
Substrate
n/a
Meas. Tech.
ChEMBL_810654 (CHEMBL2015705)
IC50
8±n/a nM
Citation
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More Info.:
Target
Name:
Tyrosine-protein kinase Blk
Synonyms:
B lymphocyte kinase | BLK_MOUSE | Blk | p55-Blk
Type:
PROTEIN
Mol. Mass.:
56676.10
Organism:
Mus musculus
Description:
ChEMBL_810654
Residue:
499
Sequence:
MGLLSSKRQVSEKGKGWSPVKIRTQDKAPPPLPPLVVFNHLAPPSPNQDPDEEERFVVALFDYAAVNDRDLQVLKGEKLQVLRSTGDWWLARSLVTGREGYVPSNFVAPVETLEVEKWFFRTISRKDAERQLLAPMNKAGSFLIRESESNKGAFSLSVKDITTQGEVVKHYKIRSLDNGGYYISPRITFPTLQALVQHYSKKGDGLCQKLTLPCVNLAPKNLWAQDEWEIPRQSLKLVRKLGSGQFGEVWMGYYKNNMKVAIKTLKEGTMSPEAFLGEANVMKTLQHERLVRLYAVVTREPIYIVTEYMARGCLLDFLKTDEGSRLSLPRLIDMSAQVAEGMAYIERMNSIHRDLRAANILVSETLCCKIADFGLARIIDSEYTAQEGAKFPIKWTAPEAIHFGVFTIKADVWSFGVLLMEIVTYGRVPYPGMSNPEVIRSLEHGYRMPCPETCPPELYNDIITECWRGRPEERPTFEFLQSVLEDFYTATEGQYELQP