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Target
Vasoactive intestinal polypeptide receptor 2
Ligand
BDBM50445114
Substrate
n/a
Meas. Tech.
ChEMBL_1284427 (CHEMBL3106155)
EC50
0.39±n/a nM
Citation
 Giordanetto, F; Revell, JD; Knerr, L; Hostettler, M; Paunovic, A; Priest, C; Janefeldt, A; Gill, A Stapled Vasoactive Intestinal Peptide (VIP) Derivatives Improve VPAC2 Agonism and Glucose-Dependent Insulin Secretion. ACS Med Chem Lett 4:1163-8 (2013) [PubMed]  Article 
Target
Name:
Vasoactive intestinal polypeptide receptor 2
Synonyms:
VIP 2 | VIP2R | VIPR2 | VIPR2_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49488.30
Organism:
Homo sapiens (Human)
Description:
VIP 2 VIPR2 HUMAN::P41587
Residue:
438
Sequence:
MRTLLPPALLTCWLLAPVNSIHPECRFHLEIQEEETKCAELLRSQTEKHKACSGVWDNITCWRPANVGETVTVPCPKVFSNFYSKAGNISKNCTSDGWSETFPDFVDACGYSDPEDESKITFYILVKAIYTLGYSVSLMSLATGSIILCLFRKLHCTRNYIHLNLFLSFILRAISVLVKDDVLYSSSGTLHCPDQPSSWVGCKLSLVFLQYCIMANFFWLLVEGLYLHTLLVAMLPPRRCFLAYLLIGWGLPTVCIGAWTAARLYLEDTGCWDTNDHSVPWWVIRIPILISIIVNFVLFISIIRILLQKLTSPDVGGNDQSQYKRLAKSTLLLIPLFGVHYMVFAVFPISISSKYQILFELCLGSFQGLVVAVLYCFLNSEVQCELKRKWRSRCPTPSASRDYRVCGSSFSRNGSEGALQFHRGSRAQSFLQTETSVI
  
Inhibitor
Name:
BDBM50445114
Synonyms:
CHEMBL3105020
Type:
Small organic molecule
Emp. Form.:
C164H268N44O43
Mol. Mass.:
3544.1517
SMILES:
n/a
Structure:
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