Reaction Details Report a problem with these data
Target
Formyl peptide receptor-related sequence 1
Ligand
BDBM50097563
Substrate
n/a
Meas. Tech.
ChEMBL_1504350 (CHEMBL3592687)
EC50
2500±n/a nM
Citation
Lacivita, E; Schepetkin, IA; Stama, ML; Kirpotina, LN; Colabufo, NA; Perrone, R; Khlebnikov, AI; Quinn, MT; Leopoldo, M Novel 3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamides as selective agonists of human formyl-peptide receptor 2. Bioorg Med Chem 23:3913-24 (2015) [PubMed] Article
More Info.:
Target
Name:
Formyl peptide receptor-related sequence 1
Synonyms:
FMLP-R-I | FMLP-related receptor I | FPRS1_MOUSE | Formyl peptide receptor related sequence 1 | Formyl peptide receptor-like 1 | Fpr-s1 | Fpr2 | Fpr3 | Fprl1 | LXA4 receptor | Lipoxin A4 receptor | Lxa4r | N-formyl peptide receptor 2 | N-formyl peptide receptor 3
Type:
PROTEIN
Mol. Mass.:
39532.25
Organism:
Mouse
Description:
ChEMBL_109574
Residue:
351
Sequence:
METNYSIPLNGSDVVIYDSTISRVLWILSMVVVSITFFLGVLGNGLVIWVAGFRMPHTVTTIWYLNLALADFSFTATLPFLLVEMAMKEKWPFGWFLCKLVHIAVDVNLFGSVFLIAVIALDRCICVLHPVWAQNHRTVSLARNVVVGSWIFALILTLPLFLFLTTVRDARGDVHCRLSFVSWGNSVEERLNTAITFVTTRGIIRFIVSFSLPMSFVAICYGLITTKIHKKAFVNSSRPFRVLTGVVASFFICWFPFQLVALLGTVWLKEMQFSGSYKIIGRLVNPTSSLAFFNSCLNPILYVFMGQDFQERLIHSLSSRLQRALSEDSGHISDTRTNLASLPEDIEIKAI