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Target
Chromobox protein homolog 5
Ligand
BDBM50194471
Substrate
n/a
Meas. Tech.
ChEMBL_1616626 (CHEMBL3858695)
IC50
26000±n/a nM
Citation
Stuckey, JI; Simpson, C; Norris-Drouin, JL; Cholensky, SH; Lee, J; Pasca, R; Cheng, N; Dickson, BM; Pearce, KH; Frye, SV; James, LI Structure-Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains. J Med Chem 59:8913-8923 (2016) [PubMed] Article
More Info.:
Target
Name:
Chromobox protein homolog 5
Synonyms:
Antigen p25 | CBX5 | CBX5_HUMAN | Chromobox protein homolog 5 | HP1 alpha | HP1A | Heterochromatin protein 1 homolog alpha
Type:
PROTEIN
Mol. Mass.:
22222.71
Organism:
Human
Description:
ChEMBL_116826
Residue:
191
Sequence:
MGKKTKRTADSSSSEDEEEYVVEKVLDRRVVKGQVEYLLKWKGFSEEHNTWEPEKNLDCPELISEFMKKYKKMKEGENNKPREKSESNKRKSNFSNSADDIKSKKKREQSNDIARGFERGLEPEKIIGATDSCGDLMFLMKWKDTDEADLVLAKEANVKCPQIVIAFYEERLTWHAYPEDAENKEKETAKS