Reaction Details
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Target
Potassium voltage-gated channel subfamily A member 1
Ligand
BDBM50237157
Substrate
n/a
Meas. Tech.
ChEMBL_1659946 (CHEMBL4009558)
IC50
14000±n/a nM
Citation
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More Info.:
Target
Name:
Potassium voltage-gated channel subfamily A member 1
Synonyms:
KCNA1_RAT | Kcna1 | Potassium voltage-gated channel subfamily A member 1 | RBKI | RCK1 | Voltage-gated potassium channel subunit Kv1.1
Type:
PROTEIN
Mol. Mass.:
56364.13
Organism:
Rattus norvegicus
Description:
ChEMBL_117743
Residue:
495
Sequence:
MTVMSGENADEASAAPGHPQDGSYPRQADHDDHECCERVVINISGLRFETQLKTLAQFPNTLLGNPKKRMRYFDPLRNEYFFDRNRPSFDAILYYYQSGGRLRRPVNVPLDMFSEEIKFYELGEEAMEKFREDEGFIKEEERPLPEKEYQRQVWLLFEYPESSGPARVIAIVSVMVILISIVIFCLETLPELKDDKDFTGTIHRIDNTTVIYTSNIFTDPFFIVETLCIIWFSFELVVRFFACPSKTDFFKNIMNFIDIVAIIPYFITLGTEIAEQEGNQKGEQATSLAILRVIRLVRVFRIFKLSRHSKGLQILGQTLKASMRELGLLIFFLFIGVILFSSAVYFAEAEEAESHFSSIPDAFWWAVVSMTTVGYGDMYPVTIGGKIVGSLCAIAGVLTIALPVPVIVSNFNYFYHRETEGEEQAQLLHVSSPNLASDSDLSRRSSSTISKSEYMEIEEDMNNSIAHYRQANIRTGNCTATDQNCVNKSKLLTDV