Reaction Details Report a problem with these data
Target
Histamine H2 receptor
Ligand
BDBM82472
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_456
Citation
Kennett, GA; Bright, F; Trail, B; Baxter, GS; Blackburn, TP Effects of the 5-HT2B receptor agonist, BW 723C86, on three rat models of anxiety. Br J Pharmacol 117:1443-8 (1996) [PubMed] Article
More Info.:
Target
Name:
Histamine H2 receptor
Synonyms:
HISTAMINE H2 | HRH2_MOUSE | Hrh2 | Hrh2 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
44816.27
Organism:
Mouse
Description:
P97292
Residue:
397
Sequence:
MEPNGTVHSCCLDSIALKVTISVVLTTLIFITVAGNVVVCLAVSLNRRLRSLTNCFIVSLAATDLLLGLLVMPFSAIYQLSFKWSFGQVFCNIYTSLDVMLCTASILNLFMISLDRYCAVTDPLRYPVLVTPVRVAISLVFIWVISITLSFLSIHLGWNSRNGTRGGNDTFKCKVQVNEVYGLVDGMVTFYLPLLIMCVTYYRIFKIAREQAKRINHISSWKAATIREHKATVTLAAVMGAFIVCWFPYFTAFVYRGLRGDDAVNEVVEGIVLWLGYANSALNPILYATLNRDFRMAYQQLFHCKLASHNSHKTSLRLNNSLLSRSQSREGRWQEEKPLKLQVWSGTELTHPQGSPVRTRLSHSSCLLSLSLLSFIWKLGTWIHHRRPFQPSLHISA