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Target
Histamine H4 receptor
Ligand
BDBM7966
Substrate
n/a
Ki
17±n/a nM
Comments
PDSP_934
Citation
Zhu, Y; Michalovich, D; Wu, H; Tan, KB; Dytko, GM; Mannan, IJ; Boyce, R; Alston, J; Tierney, LA; Li, X; Herrity, NC; Vawter, L; Sarau, HM; Ames, RS; Davenport, CM; Hieble, JP; Wilson, S; Bergsma, DJ; Fitzgerald, LR Cloning, expression, and pharmacological characterization of a novel human histamine receptor. Mol Pharmacol 59:434-41 (2001) [PubMed] Article
More Info.:
Target
Name:
Histamine H4 receptor
Synonyms:
AXOR35 | G-protein coupled receptor 105 | GPCR105 | GPRv53 | HH4R | HISTAMINE H4 | HRH4 | HRH4_HUMAN | Histamine H4 receptor | Histamine H4 receptor (H4R) | Histamine receptor (H3 and H4) | Pfi-013 | SP9144
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44517.02
Organism:
Human
Description:
Binding assays were using CHO cells stably expressing hH4R receptors.
Residue:
390
Sequence:
MPDTNSTINLSLSTRVTLAFFMSLVAFAIMLGNALVILAFVVDKNLRHRSSYFFLNLAISDFFVGVISIPLYIPHTLFEWDFGKEICVFWLTTDYLLCTASVYNIVLISYDRYLSVSNAVSYRTQHTGVLKIVTLMVAVWVLAFLVNGPMILVSESWKDEGSECEPGFFSEWYILAITSFLEFVIPVILVAYFNMNIYWSLWKRDHLSRCQSHPGLTAVSSNICGHSFRGRLSSRRSLSASTEVPASFHSERQRRKSSLMFSSRTKMNSNTIASKMGSFSQSDSVALHQREHVELLRARRLAKSLAILLGVFAVCWAPYSLFTIVLSFYSSATGPKSVWYRIAFWLQWFNSFVNPLLYPLCHKRFQKAFLKIFCIKKQPLPSQHSRSVSS