Reaction Details Report a problem with these data
Target
Peptidyl-prolyl cis-trans isomerase C
Ligand
BDBM92912
Substrate
n/a
Meas. Tech.
PPIase Assay
pH
7.8±n/a
Temperature
278.15±n/a K
Ki
>1.00e+5±n/a nM
Comments
extracted
Citation
Daum, S; Schumann, M; Mathea, S; Aumüller, T; Balsley, MA; Constant, SL; de Lacroix, BF; Kruska, F; Braun, M; Schiene-Fischer, C Isoform-specific inhibition of cyclophilins. Biochemistry 48:6268-77 (2009) [PubMed] Article
More Info.:
Target
Name:
Peptidyl-prolyl cis-trans isomerase C
Synonyms:
CYPC | Cyclophilin C (CypC) | PPIC | PPIC_HUMAN | Peptidyl-prolyl cis-trans isomerase C
Type:
Protein
Mol. Mass.:
22767.52
Organism:
Human
Description:
P45877
Residue:
212
Sequence:
MGPGPRLLLPLVLCVGLGALVFSSGAEGFRKRGPSVTAKVFFDVRIGDKDVGRIVIGLFGKVVPKTVENFVALATGEKGYGYKGSKFHRVIKDFMIQGGDITTGDGTGGVSIYGETFPDENFKLKHYGIGWVSMANAGPDTNGSQFFITLTKPTWLDGKHVVFGKVIDGMTVVHSIELQATDGHDRPLTNCSIINSGKIDVKTPFVVEIADW