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Target
Guanine nucleotide-binding protein subunit alpha-15
Ligand
BDBM96792
Substrate
n/a
EC50
19414±n/a nM
Citation
 PubChem, PC Counterscreen for agonists of the human trace amine associated receptor 1 (TAAR1): Fluorescence-based cell-based high throughput dose response assay to identify nonselective Ga16 agonists PubChem Bioassay (2013)[AID] 
Target
Name:
Guanine nucleotide-binding protein subunit alpha-15
Synonyms:
G protein alpha 16 | G-protein subunit alpha-16 | G-protein subunit alpha-16 (G alpha-16) | GNA15 | GNA15_HUMAN | GNA16 | Guanine nucleotide-binding protein subunit alpha-15 [Y147C]
Type:
Protein
Mol. Mass.:
43577.62
Organism:
Human
Description:
P30679
Residue:
374
Sequence:
MARSLTWRCCPWCLTEDEKAAARVDQEINRILLEQKKQDRGELKLLLLGPGESGKSTFIKQMRIIHGAGYSEEERKGFRPLVYQNIFVSMRAMIEAMERLQIPFSRPESKHHASLVMSQDPYKVTTFEKRYAAAMQWLWRDAGIRACYERRREFHLLDSAVYYLSHLERITEEGYVPTAQDVLRSRMPTTGINEYCFSVQKTNLRIVDVGGQKSERKKWIHCFENVIALIYLASLSEYDQCLEENNQENRMKESLALFGTILELPWFKSTSVILFLNKTDILEEKIPTSHLATYFPSFQGPKQDAEAAKRFILDMYTRMYTGCVDGPEGSKKGARSRRLFSHYTCATDTQNIRKVFKDVRDSVLARYLDEINLL
  
Inhibitor
Name:
BDBM96792
Synonyms:
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-(3-ethoxyphenyl)-N-[(E)-(5-methyl-2-furanyl)methylideneamino]-4-triazolecarboxamide | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-(3-ethoxyphenyl)-N-[(E)-(5-methylfuran-2-yl)methylideneamino]triazole-4-carboxamide | 1-(4-aminofurazan-3-yl)-N-[(E)-(5-methyl-2-furyl)methyleneamino]-5-m-phenetyl-triazole-4-carboxamide | 1-(4-azanyl-1,2,5-oxadiazol-3-yl)-5-(3-ethoxyphenyl)-N-[(E)-(5-methylfuran-2-yl)methylideneamino]-1,2,3-triazole-4-carboxamide | MLS001142536 | SMR000647884 | cid_9631625
Type:
Small organic molecule
Emp. Form.:
C19H18N8O4
Mol. Mass.:
422.3974
SMILES:
CCOc1cccc(c1)-c1c(nnn1-c1nonc1N)C(=O)N\N=C\c1ccc(C)o1
Structure:
Search PDB for entries with ligand similarity: