Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM46392
Substrate
n/a
IC50
2267±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Homo sapiens (Human)
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM46392
Synonyms:
2-[(4-propoxybenzyl)thio]-1H-benzimidazole | 2-[(4-propoxyphenyl)methylsulfanyl]-1H-benzimidazole | 2-[(4-propoxyphenyl)methylthio]-1H-benzimidazole | MLS000577054 | SMR000198134 | cid_1653621
Type:
Small organic molecule
Emp. Form.:
C17H18N2OS
Mol. Mass.:
298.403
SMILES:
CCCOc1ccc(CSc2nc3ccccc3[nH]2)cc1
Structure:
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