Reaction Details Report a problem with these data
Target
Mitogen-activated protein kinase 1 [L198A,L232A]
Ligand
BDBM176676
Substrate
n/a
Meas. Tech.
Fluorescence Quenching Assay
Kd
140±20 nM
Citation
Shapiro, PS; MacKerell, Jr., AD; Fletcher, S Non-ATP dependent inhibitors of extracellular signal-regulated kinase (ERK) US Patent US9115122 Publication Date 8/25/2015
More Info.:
Target
Name:
Mitogen-activated protein kinase 1 [L198A,L232A]
Synonyms:
ERK2(L198A/L232A) | Erk2 | MK01_MOUSE | Mapk | Mapk1 | Prkm1
Type:
n/a
Mol. Mass.:
41194.49
Organism:
Mouse
Description:
P63085[L198A,L232A]
Residue:
358
Sequence:
MAAAAAAGPEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNLNKVRVAIKKISPFEHQTYCQRTLREIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFLYQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVATRWYRAPEIMANSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYADQLNHILGILGSPSQEDLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAHPYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGYRS