Reaction Details Report a problem with these data
Target
Adenosine receptor A3 [I248L]
Ligand
BDBM191052
Substrate
n/a
Meas. Tech.
Radioligand Binding Assay
pH
7.5±n/a
Temperature
298.15±n/a K
Ki
1530±60 nM
Comments
extracted
Citation
Jacobson, KA; Tosh, DK Adenosine receptor agonists, partial agonists, and antagonists US Patent US9181253 Publication Date 11/10/2015
More Info.:
Target
Name:
Adenosine receptor A3 [I248L]
Synonyms:
AA3R_HUMAN | ADORA3 | Adenosine receptor A3 | Adenosine receptor A3 (A3)
Type:
Protein
Mol. Mass.:
36197.32
Organism:
Human
Description:
P0DMS8[I248L]
Residue:
318
Sequence:
MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKRVTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYFSFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFALSWLPLSLINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKACVVCHPSDSLDTSIEKNSE