Reaction Details Report a problem with these data
Target
WD repeat-containing protein 5 [24-334]
Ligand
BDBM200659
Substrate
n/a
Meas. Tech.
Binding Assay
pH
6.5±n/a
Temperature
298.15±n/a K
IC50
<100±n/a nM
Comments
extracted
Citation
Wang, S; Karatas, H; Dou, Y; Townsend, E; Bernard, D Inhibition of WDR5 interaction with its binding partners US Patent US9233086 Publication Date 1/12/2016
More Info.:
Target
Name:
WD repeat-containing protein 5 [24-334]
Synonyms:
BIG3 | WD repeat-containing protein 5 (WDR5) | WDR5 | WDR5_HUMAN
Type:
n/a
Mol. Mass.:
34198.55
Organism:
Human
Description:
N-terminal His-tagged WDR5Delta23 (residues 24-334)
Residue:
311
Sequence:
TQSKPTPVKPNYALKFTLAGHTKAVSSVKFSPNGEWLASSSADKLIKIWGAYDGKFEKTISGHKLGISDVAWSSDSNLLVSASDDKTLKIWDVSSGKCLKTLKGHSNYVFCCNFNPQSNLIVSGSFDESVRIWDVKTGKCLKTLPAHSDPVSAVHFNRDGSLIVSSSYDGLCRIWDTASGQCLKTLIDDDNPPVSFVKFSPNGKYILAATLDNTLKLWDYSKGKCLKTYTGHKNEKYCIFANFSVTGGKWIVSGSEDNLVYIWNLQTKEIVQKLQGHTDVVISTACHPTENIIASAALENDKTIKLWKSDC