Reaction Details Report a problem with these data
Target
Inorganic pyrophosphatase
Ligand
BDBM205469
Substrate
n/a
Meas. Tech.
Colorimetric Malachite Green Assay
pH
7.5±n/a
Temperature
298.15±n/a K
IC50
9.82e+4± 8e+3 nM
Comments
extracted
Citation
Pang, AH; Garzan, A; Larsen, MJ; McQuade, TJ; Garneau-Tsodikova, S; Tsodikov, OV Discovery of Allosteric and Selective Inhibitors of Inorganic Pyrophosphatase from Mycobacterium tuberculosis. ACS Chem Biol 11:3084-3092 (2016) [PubMed] Article
More Info.:
Target
Name:
Inorganic pyrophosphatase
Synonyms:
IPYR_ECOLI | Inorganic pyrophosphatase (EcPPiase) | ppa
Type:
Protein
Mol. Mass.:
19696.77
Organism:
Escherichia coli (strain K12)
Description:
P0A7A9
Residue:
176
Sequence:
MSLLNVPAGKDLPEDIYVVIEIPANADPIKYEIDKESGALFVDRFMSTAMFYPCNYGYINHTLSLDGDPVDVLVPTPYPLQPGSVIRCRPVGVLKMTDEAGEDAKLVAVPHSKLSKEYDHIKDVNDLPELLKAQIAHFFEHYKDLEKGKWVKVEGWENAEAAKAEIVASFERAKNK