Reaction Details
Report a problem with these data
![](/images/Email.png)
Target
Kappa-type opioid receptor [Y66A]
Ligand
BDBM214799
Substrate
n/a
Meas. Tech.
cAMP Inhibition Assay
pH
7.4±n/a
EC50
1.5e+2±1e+1 nM
Comments
extracted
Citation
![](/images/small/blackdot.gif)
More Info.:
Target
Name:
Kappa-type opioid receptor [Y66A]
Synonyms:
Kappa opioid receptor (KOR Y66A) | OPRK | OPRK1 | OPRK_HUMAN
Type:
Protein
Mol. Mass.:
42556.66
Organism:
Homo sapiens (Human)
Description:
Human KOR with Y66A mutation
Residue:
380
Sequence:
MDSPIQIFRGEPGPTCAPSACLPPNSSAWFPGWAEPDSNGSAGSEDAQLEPAHISPAIPVIITAVASVVFVVGLVGNSLVMFVIIRYTKMKTATNIYIFNLALADALVTTTMPFQSTVYLMNSWPFGDVLCKIVISIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPLKAKIINICIWLLSSSVGISAIVLGGTKVREDVDVIECSLQFPDDDYSWWDLFMKICVFIFAFVIPVLIIIVCYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFVVCWTPIHIFILVEALGSTSHSTAALSSYYFCIALGYTNSSLNPILYAFLDENFKRCFRDFCFPLKMRMERQSTSRVRNTVQDPAYLRDIDGMNKPV