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Target
Proto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C]
Ligand
BDBM234844
Substrate
n/a
Meas. Tech.
In vitro Kinase Assay
pH
8±n/a
IC50
29±n/a nM
Comments
extracted
Citation
Garske, AL; Shokat, KM Methods and compositions for kinase inhibition US Patent US9353116 Publication Date 5/31/2016
More Info.:
Target
Name:
Proto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C]
Synonyms:
Proto-oncogene tyrosine-protein kinase Src (T338C/V323S) | SRC | SRC_CHICK
Type:
Protein
Mol. Mass.:
32350.41
Organism:
Chicken
Description:
residues 251-533
Residue:
283
Sequence:
QTQGLAKDAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLSQLYAVVSEEPIYIVCEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLIEDNEYTARQGAKFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL