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Target
Serine/threonine-protein kinase Nek2 [T175A]
Ligand
BDBM259826
Substrate
n/a
Meas. Tech.
Nek2 Inhibition Assay
pH
7.6±n/a
Temperature
298.15±n/a K
IC50
>300000±n/a nM
Comments
extracted
Citation
Taunton, Jr., JW; Maglathlin, R; Serafimova, I; Cohen, MS; Miller, R; Paavilainen, V; McFarland, J; Krishnan, S Kinase inhibitors US Patent US9505766 Publication Date 11/29/2016
More Info.:
Target
Name:
Serine/threonine-protein kinase Nek2 [T175A]
Synonyms:
NEK2 | NEK2A | NEK2_HUMAN | NLK1 | Serine/threonine-protein kinase Nek2 (T175A)
Type:
Enzyme
Mol. Mass.:
51746.94
Organism:
Human
Description:
Full-length human T175A NEK2 (referred to as "NEK2").
Residue:
445
Sequence:
MPSRAEDYEVLYTIGTGSYGRCQKIRRKSDGKILVWKELDYGSMTEAEKQMLVSEVNLLRELKHPNIVRYYDRIIDRTNTTLYIVMEYCEGGDLASVITKGTKERQYLDEEFVLRVMTQLTLALKECHRRSDGGHTVLHRDLKPANVFLDGKQNVKLGDFGLARILNHDTSFAKAFVGTPYYMSPEQMNRMSYNEKSDIWSLGCLLYELCALMPPFTAFSQKELAGKIREGKFRRIPYRYSDELNEIITRMLNLKDYHRPSVEEILENPLIADLVADEQRRNLERRGRQLGEPEKSQDSSPVLSELKLKEIQLQERERALKAREERLEQKEQELCVRERLAEDKLARAENLLKNYSLLKERKFLSLASNPELLNLPSSVIKKKVHFSGESKENIMRSENSESQLTSKSKCKDLKKRLHAAQLRAQALSDIEKNYQLKSRQILGMR