Reaction Details Report a problem with these data
Target
Endothelin-1
Ligand
BDBM172573
Substrate
n/a
Meas. Tech.
ET-1 Assay
EC50
<50000±n/a nM
Citation
PubChem, PC; Buckman, BO; Nicholas, JB; Ramphal, JY; Emayan, K; Seiwert, SD Anti-fibrotic pyridinones US Patent US9675593 Publication Date 6/13/2017
More Info.:
Target
Name:
Endothelin-1
Synonyms:
EDN1 | EDN1_HUMAN | PPET1 | Preproendothelin-1
Type:
Protein
Mol. Mass.:
24444.51
Organism:
Human
Description:
P05305
Residue:
212
Sequence:
MDYLLMIFSLLFVACQGAPETAVLGAELSAVGENGGEKPTPSPPWRLRRSKRCSCSSLMDKECVYFCHLDIIWVNTPEHVVPYGLGSPRSKRALENLLPTKATDRENRCQCASQKDKKCWNFCQAGKELRAEDIMEKDWNNHKKGKDCSKLGKKCIYQQLVRGRKIRRSSEEHLRQTRSETMRNSVKSSFHDPKLKGKPSRERYVTHNRAHW