Reaction Details Report a problem with these data
Target
Botulinum neurotoxin type A [1-429]
Ligand
BDBM506808
Substrate
n/a
Meas. Tech.
BoNT/A LC429 Enzymatic assay
Ki
6.40±n/a nM
Citation
Jiao, G; Johnson, AT; O''Malley, S; Kim, SJ Hydroxamic acids comprising pyrazole moiety and uses thereof US Patent US11046652 Publication Date 6/29/2021
More Info.:
Target
Name:
Botulinum neurotoxin type A [1-429]
Synonyms:
BXA1_CLOBH | BoNT/A LC | Botulinum neurotoxin type A | bna | botA
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49198.33
Organism:
Clostridium botulinum (strain Hall / ATCC 3502 / NCTC 13319 / Type A)
Description:
P0DPI1[1-429] First 11 removed
Residue:
429
Sequence:
MPFVNKQFNYKDPVNGVDIAYIKIPNAGQMQPVKAFKIHNKIWVIPERDTFTNPEEGDLNPPPEAKQVPVSYYDSTYLSTDNEKDNYLKGVTKLFERIYSTDLGRMLLTSIVRGIPFWGGSTIDTELKVIDTNCINVIQPDGSYRSEELNLVIIGPSADIIQFECKSFGHEVLNLTRNGYGSTQYIRFSPDFTFGFEESLEVDTNPLLGAGKFATDPAVTLAHELIHAGHRLYGIAINPNRVFKVNTNAYYEMSGLEVSFEELRTFGGHDAKFIDSLQENEFRLYYYNKFKDIASTLNKAKSIVGTTASLQYMKNVFKEKYLLSEDTSGKFSVDKLKFDKLYKMLTEIYTEDNFVKFFKVLNRKTYLNFDKAVFKINIVPKVNYTIYDGFNLRNTNLAANFNGQNTEINNMNFTKLKNFTGLFEFYKLL