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Target
Bromodomain-containing protein 4 [44-167]
Ligand
BDBM550488
Substrate
n/a
Meas. Tech.
ATPLITE assay
IC50
53.0±n/a nM
Citation
Bradner, JE; Qi, J; Tanaka, M; Buckley, D Cyano thienotriazolodiazepines and uses thereof US Patent US11306105 Publication Date 4/19/2022
More Info.:
Target
Name:
Bromodomain-containing protein 4 [44-167]
Synonyms:
BRD4 | BRD4 bromodomain 1 | BRD4_HUMAN | Brd4-1 | HUNK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
14738.39
Organism:
Homo sapiens (Human)
Description:
O60885[44-167]
Residue:
124
Sequence:
NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTE