Reaction Details Report a problem with these data
Target
Stimulator of interferon genes protein [1-379,R71H,G230A,H232R,R293Q]
Ligand
BDBM550796
Substrate
n/a
Meas. Tech.
H-cGAMP Filtration Binding Assay (HAQ STING)
IC50
1216±n/a nM
Citation
Altman, MD; Childers, ML; Jewell, JP; Lesburg, CA; Siu, T Oxo-tetrahydro-isoquinoline carboxylic acids as STING inhibitors US Patent US11311528 Publication Date 4/26/2022
More Info.:
Target
Name:
Stimulator of interferon genes protein [1-379,R71H,G230A,H232R,R293Q]
Synonyms:
ERIS | HAQ STING(1-379) (R71H, G230A, H232R, R293Q) | MITA | STING | STING1 | STING_HUMAN | Stimulator of interferon genes protein (1-379) (R71H, G230A, H232R, R293Q) | Stimulator of interferon genes protein [R71H,G230A,H232R,R293Q] | TMEM173
Type:
Protein
Mol. Mass.:
42180.60
Organism:
Human
Description:
HAQ STING(1-379) (R71H, G230A, H232R, R293Q)
Residue:
379
Sequence:
MPHSSLHPSIPCPRGHGAQKAALVLLSACLVTLWGLGEPPEHTLRYLVLHLASLQLGLLLNGVCSLAEELHHIHSRYRGSYWRTVRACLGCPLRRGALLLLSIYFYYSLPNAVGPPFTWMLALLGLSQALNILLGLKGLAPAEISAVCEKGNFNVAHGLAWSYYIGYLRLILPELQARIRTYNQHYNNLLRGAVSQRLYILLPLDCGVPDNLSMADPNIRFLDKLPQQTADRAGIKDRVYSNSIYELLENGQRAGTCVLEYATPLQTLFAMSQYSQAGFSREDRLEQAKLFCQTLEDILADAPESQNNCRLIAYQEPADDSSFSLSQEVLRHLRQEEKEEVTVGSLKTSAVPSTSTMSQEPELLISGMEKPLPLRTDFS