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Target
Somatostatin receptor type 1
Ligand
BDBM311911
Substrate
n/a
Meas. Tech.
Binding Assay
Ki
>9148±n/a nM
Citation
 Coates, DA; Remick, DM SSTR4 agonist salts US Patent  US11834435 Publication Date 12/5/2023 
Target
Name:
Somatostatin receptor type 1
Synonyms:
SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1)
Type:
Enzyme
Mol. Mass.:
42692.81
Organism:
Homo sapiens (Human)
Description:
P30872
Residue:
391
Sequence:
MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAILISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLLRHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLGVWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAICLCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQDDATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKSRAYSVEDFQPENLESGGVFRNGTCTSRITTL
  
Inhibitor
Name:
BDBM311911
Synonyms:
US10166214, Example 47 | US10675268, Example 47 | US11834435, Example 3 | US9789082, Example 47
Type:
Small organic molecule
Emp. Form.:
C16H23N3O2
Mol. Mass.:
289.3727
SMILES:
Cc1cccnc1OCC(C)(C)NC(=O)[C@@H]1[C@H]2CNC[C@@H]12 |r|
Structure:
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