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Target
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
Ligand
BDBM347359
Substrate
n/a
Meas. Tech.
In Vitro Assay
IC50
2.74±n/a nM
Citation
Markowitz, S; Willson, JK; Posner, B; Ready, J; Antczak, M; Zhang, Y; Desai, A; Gerson, S; Greenlee, W Compositions and methods of modulating short-chain dehydrogenase activity US Patent US9789116 Publication Date 10/17/2017
More Info.:
Target
Name:
15-hydroxyprostaglandin dehydrogenase [NAD(+)]
Synonyms:
15-PGDH | Hpgd | PGDH_RAT | Pgdh1 | Prostaglandin dehydrogenase 1 (15-PGDH)
Type:
Protein
Mol. Mass.:
28938.62
Organism:
Rattus norvegicus (Rat)
Description:
O08699
Residue:
266
Sequence:
MHVNGKVALVTGAAQGIGKAFTEALLLHGAKVALVDWNLETGVKCKAALDEQFEPQKTLFIQCDVADQKQLRDTFRKVVDHFGRLDILVNNAGVNNEKNWEQTLQINLVSVISGTYLGLDYMSKQNGGEGGIIINISSIAGLMPVAQQPVYCASKHGIIGFTRSAAMAANLMKSGVRLNVICPGFVKTPILESIEKEENMGQYIEYTDQIKAMMKFYGILDPSAIANGLINLIEDDALNGAIMKITASKGIHFQDYDLFPSFSKAP