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Target
MAP kinase-interacting serine/threonine-protein kinase 1 [1-424]
Ligand
BDBM227728
Substrate
n/a
Meas. Tech.
MKNK1 Kinase High ATP Assay
pH
7.5±n/a
IC50
2±n/a nM
Comments
extracted
Citation
Klar, U; Wortmann, L; Kettschau, G; Pühler, F; Lienau, P; Sülzle, D Substituted pyrazolopyrimidinylamino-indazoles US Patent US9556181 Publication Date 1/31/2017
More Info.:
Target
Name:
MAP kinase-interacting serine/threonine-protein kinase 1 [1-424]
Synonyms:
MAP kinase signal-integrating kinase 1 (MKNK1) | MKNK1 | MKNK1_HUMAN | MNK1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47005.82
Organism:
Homo sapiens (Human)
Description:
aa 1-424
Residue:
424
Sequence:
MVSSQKLEKPIEMGSSEPLPIADGDRRRKKKRRGRATDSLPGKFEDMYKLTSELLGEGAYAKVQGAVSLQNGKEYAVKIIEKQAGHSRSRVFREVETLYQCQGNKNILELIEFFEDDTRFYLVFEKLQGGSILAHIQKQKHFNEREASRVVRDVAAALDFLHTKDKVSLCHLGWSAMAPSGLTAAPTSLGSSDPPTSASQVAGTTGIAHRDLKPENILCESPEKVSPVKICDFDLGSGMKLNNSCTPITTPELTTPCGSAEYMAPEVVEVFTDQATFYDKRCDLWSLGVVLYIMLSGYPPFVGHCGADCGWDRGEVCRVCQNKLFESIQEGKYEFPDKDWAHISSEAKDLISKLLVRDAKQRLSAAQVLQHPWVQGQAPEKGLPTPQVLQRNSSTMDLTLFAAEAIALNRQLSQHEENELAEEP