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Target
P2Y purinoceptor 13
Ligand
BDBM359084
Substrate
n/a
Meas. Tech.
Ca++ flux assay
EC50
42370000±n/a nM
Citation
 Dasseux, JH; Barbaras, R Compounds, compositions and methods useful for cholesterol mobilization US Patent  US10220040 Publication Date 3/5/2019 
Target
Name:
P2Y purinoceptor 13
Synonyms:
G-protein coupled receptor 86 | G-protein coupled receptor 94 | GPR86 | GPR94 | P2RY13 | P2Y13 | P2Y13_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40817.42
Organism:
Homo sapiens (Human)
Description:
n/a
Residue:
354
Sequence:
MTAAIRRQRELSILPKVTLEAMNTTVMQGFNRSERCPRDTRIVQLVFPALYTVVFLTGILLNTLALWVFVHIPSSSTFIIYLKNTLVADLIMTLMLPFKILSDSHLAPWQLRAFVCRFSSVIFYETMYVGIVLLGLIAFDRFLKIIRPLRNIFLKKPVFAKTVSIFIWFFLFFISLPNTILSNKEATPSSVKKCASLKGPLGLKWHQMVNNICQFIFWTVFILMLVFYVVIAKKVYDSYRKSKSKDRKNNKKLEGKVFVVVAVFFVCFAPFHFARVPYTHSQTNNKTDCRLQNQLFIAKETTLFLAATNICMDPLIYIFLCKKFTEKLPCMQGRKTTASSQENHSSQTDNITLG
  
Inhibitor
Name:
BDBM359084
Synonyms:
US10220040, Compound Ih-(R-isomer)
Type:
Small organic molecule
Emp. Form.:
C24H32ClNO2S
Mol. Mass.:
434.034
SMILES:
CCOC(=O)C(C)(C)CCCC[C@@H](N1CCc2sccc2C1)c1ccccc1Cl |r|
Structure:
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