Reaction Details Report a problem with these data
Target
Gag-Pol polyprotein [588-1147,M628L,N654N,K657R,T802F,K807E]
Ligand
BDBM77092
Substrate
n/a
Meas. Tech.
PHENOSENSE assay
IC50
3.8±0.0 nM
Citation
Lanier, ER Methods of treating retroviral infections and related dosage regimes US Patent US9694024 Publication Date 7/4/2017
More Info.:
Target
Name:
Gag-Pol polyprotein [588-1147,M628L,N654N,K657R,T802F,K807E]
Synonyms:
HIV RT (41L/67N/70R/215F/219E) | POL_HV1H2 | gag-pol
Type:
n/a
Mol. Mass.:
64541.40
Organism:
Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)
Description:
P04585[588-1147,M628L,N654N,K657R,T802F,K807E]
Residue:
560
Sequence:
PISPIETVPVKLKPGMDGPKVKQWPLTEEKIKALVEICTELEKEGKISKIGPENPYNTPVFAIKKKNSTRWRKLVDFRELNKRTQDFWEVQLGIPHPAGLKKKKSVTVLDVGDAYFSVPLDEDFRKYTAFTIPSINNETPGIRYQYNVLPQGWKGSPAIFQSSMTKILEPFRKQNPDIVIYQYMDDLYVGSDLEIGQHRTKIEELRQHLLRWGLFTPDEKHQKEPPFLWMGYELHPDKWTVQPIVLPEKDSWTVNDIQKLVGKLNWASQIYPGIKVRQLCKLLRGTKALTEVIPLTEEAELELAENREILKEPVHGVYYDPSKDLIAEIQKQGQGQWTYQIYQEPFKNLKTGKYARMRGAHTNDVKQLTEAVQKITTESIVIWGKTPKFKLPIQKETWETWWTEYWQATWIPEWEFVNTPPLVKLWYQLEKEPIVGAETFYVDGAANRETKLGKAGYVTNRGRQKVVTLTDTTNQKTELQAIYLALQDSGLEVNIVTDSQYALGIIQAQPDQSESELVNQIIEQLIKKEKVYLAWVPAHKGIGGNEQVDKLVSAGIRKVL