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Target
Histone deacetylase 4 [627-1085]
Ligand
BDBM402284
Substrate
n/a
Meas. Tech.
Biochemical Assay
IC50
3310±n/a nM
Citation
Ma, H; Wang, Y Histone deacetylase inhibitors and methods for use thereof US Patent US10011611 Publication Date 7/3/2018
More Info.:
Target
Name:
Histone deacetylase 4 [627-1085]
Synonyms:
HDAC4 | HDAC4_HUMAN | Histone deacetylase 4 (HDAC4) (aa 627-1085) | KIAA0288
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49108.14
Organism:
Homo sapiens (Human)
Description:
aa 627-1085
Residue:
457
Sequence:
SRAQSSPASATFPVSVQEPPTKPRFTTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLNRQKLDSKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQRTTSTAGRSLIEAQTCENEEAETVTAMASLSVGVKPAEKRPDEEPMEEEPPL