Reaction Details Report a problem with these data
Target
Histone deacetylase 7 [518-592]
Ligand
BDBM402284
Substrate
n/a
Meas. Tech.
Biochemical Assay
IC50
1890±n/a nM
Citation
Ma, H; Wang, Y Histone deacetylase inhibitors and methods for use thereof US Patent US10011611 Publication Date 7/3/2018
More Info.:
Target
Name:
Histone deacetylase 7 [518-592]
Synonyms:
HDAC7 | HDAC7A | HDAC7_HUMAN | Histone deacetylase 7 (HDAC7) (aa 518-592)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47229.42
Organism:
Homo sapiens (Human)
Description:
aa 518-592
Residue:
436
Sequence:
PFTTGLIYDSVMLKHQCSCGDNSRHPEHAGRIQSIWSRLQERGLRSQCECLRGRKASLEELQSVHSERHVLLYGTNPLSRLKLDNGKLAGLLAQRMFVMLPCGGVGVDTDTIWNELHSSNAARWAAGSVTDLAFKVASRELKNGFAVVRPPGHHADHSTAMGFCFFNSVAIACRQLQQQSKASKILIVDWDVHHGNGTQQTFYQDPSVLYISLHRHDDGNFFPGSGAVDEVGAGSGEGFNVNVAWAGGLDPPMGDPEYLAAFRIVVMPIAREFSPDLVLVSAGFDAAEGHPAPLGGYHVSAKCFGYMTQQLMNLAGGAVVLALEGGHDLTAICDASEACVAALLGNRVDPLSEEGWKQKPNLNAIRSLEAVIRVHSKYWGCMQRLASCPDSWVPRVPGADKEEVEAVTALASLSVGILAEDRPSEQLVEEEEPMNL