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Target
fMet-Leu-Phe receptor
Ligand
BDBM37833
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki
>43700±n/a nM
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
fMet-Leu-Phe receptor
Synonyms:
FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38456.14
Organism:
Homo sapiens (Human)
Description:
gi_4503779
Residue:
350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVTTISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIALDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNFSPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPLRVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPMLYVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
  
Inhibitor
Name:
BDBM37833
Synonyms:
2-(2-methyl-4-oxidanylidene-7-propoxy-chromen-3-yl)isoindole-1,3-dione | 2-(2-methyl-4-oxo-7-propoxy-1-benzopyran-3-yl)isoindole-1,3-dione | 2-(2-methyl-4-oxo-7-propoxy-4H-chromen-3-yl)-1H-isoindole-1,3(2H)-dione | 2-(2-methyl-4-oxo-7-propoxychromen-3-yl)isoindole-1,3-dione | 2-(4-keto-2-methyl-7-propoxy-chromen-3-yl)isoindoline-1,3-quinone | MLS000537419 | SMR000143857 | cid_2208919
Type:
Small organic molecule
Emp. Form.:
C21H17NO5
Mol. Mass.:
363.3634
SMILES:
CCCOc1ccc2c(c1)oc(C)c(N1C(=O)c3ccccc3C1=O)c2=O
Structure:
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