Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37629
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
Ki
>40300±n/a nM
Comments
Extracted from aid = 520 and tid = 2
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37629
Synonyms:
(4E)-5-(1,3-benzodioxol-5-yl)-1-(3-methoxypropyl)-4-[oxidanyl(phenyl)methylidene]pyrrolidine-2,3-dione | (4E)-5-(1,3-benzodioxol-5-yl)-4-[hydroxy(phenyl)methylene]-1-(3-methoxypropyl)pyrrolidine-2,3-quinone | (4E)-5-(1,3-benzodioxol-5-yl)-4-[hydroxy(phenyl)methylidene]-1-(3-methoxypropyl)pyrrolidine-2,3-dione | 5-Benzo[1,3]dioxol-5-yl-4-benzoyl-3-hydroxy-1-(3-methoxy-propyl)-1,5-dihydro-pyrrol-2-one | MLS000029490 | SMR000011270 | cid_5766372
Type:
Small organic molecule
Emp. Form.:
C22H21NO6
Mol. Mass.:
395.4052
SMILES:
COCCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc2OCOc2c1
Structure:
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