Reaction Details Report a problem with these data
Target
N-formyl peptide receptor 2
Ligand
BDBM37662
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands
IC50
>66700±n/a nM
Comments
Extracted from aid = 520 and tid = 3
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor-Like-1 (FPRL1) Ligands and Dose Response Counter-Screen Assay for Formylpeptide Receptor (FPR) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
N-formyl peptide receptor 2
Synonyms:
ALXR, FPRL1, FPR2 | FMLP-related receptor I FMLP-R-I | FPR2 | FPR2_HUMAN | FPRH1 | FPRL1 | Formyl Peptide Receptor-Like 1 | HM63 | LXA4 receptor | LXA4R | Lipoxin A4 receptor | Lipoxin A4 receptor (LXA4) | RFP | hFPRL
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
38968.35
Organism:
Homo sapiens (Human)
Description:
P25090
Residue:
351
Sequence:
METNFSTPLNEYEEVSYESAGYTVLRILPLVVLGVTFVLGVLGNGLVIWVAGFRMTRTVTTICYLNLALADFSFTATLPFLIVSMAMGEKWPFGWFLCKLIHIVVDINLFGSVFLIGFIALDRCICVLHPVWAQNHRTVSLAMKVIVGPWILALVLTLPVFLFLTTVTIPNGDTYCTFNFASWGGTPEERLKVAITMLTARGIIRFVIGFSLPMSIVAICYGLIAAKIHKKGMIKSSRPLRVLTAVVASFFICWFPFQLVALLGTVWLKEMLFYGKYKIIDILVNPTSSLAFFNSCLNPMLYVFVGQDFRERLIHSLPTSLERALSEDSAPTNDTAANSASPPAETELQAM
  
Inhibitor
Name:
BDBM37662
Synonyms:
1-[2-(2-hydroxyethyloxy)ethyl]-4-oxidanyl-2-thiophen-2-yl-3-thiophen-2-ylcarbonyl-2H-pyrrol-5-one | 3-hydroxy-1-[2-(2-hydroxyethoxy)ethyl]-4-(2-thenoyl)-5-(2-thienyl)-3-pyrrolin-2-one | 4-hydroxy-1-[2-(2-hydroxyethoxy)ethyl]-3-(thiophene-2-carbonyl)-2-thiophen-2-yl-2H-pyrrol-5-one | 4-hydroxy-1-[2-(2-hydroxyethoxy)ethyl]-3-[oxo(thiophen-2-yl)methyl]-2-thiophen-2-yl-2H-pyrrol-5-one | MLS000040265 | SMR000059740 | cid_663185
Type:
Small organic molecule
Emp. Form.:
C17H17NO5S2
Mol. Mass.:
379.451
SMILES:
OCCOCCN1C(C(C(=O)c2cccs2)C(=O)C1=O)c1cccs1
Structure:
Search PDB for entries with ligand similarity: