Reaction Details Report a problem with these data
Target
Signal transducer and activator of transcription 3 [702-738,740-752]
Ligand
BDBM43617
Substrate
n/a
Meas. Tech.
Dose response cell-based assay to measure STAT3 activation
IC50
1833±n/a nM
Citation
 PubChem, PC Dose response cell-based assay to measure STAT3 activation PubChem Bioassay (2008)[AID] 
Target
Name:
Signal transducer and activator of transcription 3 [702-738,740-752]
Synonyms:
APRF | STAT3 | STAT3_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5263.93
Organism:
Homo sapiens (Human)
Description:
gi_13272532
Residue:
50
Sequence:
AAPYLKTKFICVTPTTCSNTIDLPMSPRTLDSLMQFGNGEGAEPSAGGQF
  
Inhibitor
Name:
BDBM43617
Synonyms:
MLS000583768 | N-(1H-perimidin-2-yl)benzamide | N-1H-perimidin-2-ylbenzamide | SMR000201532 | cid_1257244
Type:
Small organic molecule
Emp. Form.:
C18H13N3O
Mol. Mass.:
287.3153
SMILES:
O=C(Nc1nc2cccc3cccc([nH]1)c23)c1ccccc1
Structure:
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