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Target
Regulator of G-protein signaling 16
Ligand
BDBM47768
Substrate
n/a
Meas. Tech.
Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 16
Synonyms:
RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22748.87
Organism:
Homo sapiens (Human)
Description:
gi_156416009
Residue:
202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVLGWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEEFICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDLAAQASAASATLSSCSLDEPSHT
  
Inhibitor
Name:
BDBM47768
Synonyms:
MLS000681208 | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxy-benzamide | N-[2-(3,5-dimethylphenoxy)ethyl]-3-methoxybenzamide | SMR000269463 | cid_1562455
Type:
Small organic molecule
Emp. Form.:
C18H21NO3
Mol. Mass.:
299.3642
SMILES:
COc1cccc(c1)C(=O)NCCOc1cc(C)cc(C)c1
Structure:
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