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Target
Regulator of G-protein signaling 16
Ligand
BDBM47800
Substrate
n/a
Meas. Tech.
Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao.
EC50
>30000±n/a nM
Citation
 PubChem, PC Dose respone, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao. PubChem Bioassay (2009)[AID] 
Target
Name:
Regulator of G-protein signaling 16
Synonyms:
RGS16 | RGS16_HUMAN | RGSR | Regulator of G-protein signaling 16 (RGS16) | regulator of G-protein signalling 16
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22748.87
Organism:
Homo sapiens (Human)
Description:
gi_156416009
Residue:
202
Sequence:
MCRTLAAFPTTCLERAKEFKTRLGIFLHKSELGCDTGSTGKFEWGSKHSKENRNFSEDVLGWRESFDLLLSSKNGVAAFHAFLKTEFSEENLEFWLACEEFKKIRSATKLASRAHQIFEEFICSEAPKEVNIDHETHELTRMNLQTATATCFDAAQGKTRTLMEKDSYPRFLKSPAYRDLAAQASAASATLSSCSLDEPSHT
  
Inhibitor
Name:
BDBM47800
Synonyms:
MLS000736409 | N'-[(E)-(2-fluorophenyl)methylidene]benzenesulfonohydrazide | N-[(2-fluorobenzylidene)amino]benzenesulfonamide | N-[(2-fluorophenyl)methylideneamino]benzenesulfonamide | SMR000338359 | cid_2172475
Type:
Small organic molecule
Emp. Form.:
C13H11FN2O2S
Mol. Mass.:
278.302
SMILES:
Fc1ccccc1C=NNS(=O)(=O)c1ccccc1 |w:8.9|
Structure:
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