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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM39058
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
570±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM39058
Synonyms:
1-(4-fluorophenyl)-3-(2-hydroxy-5-methoxy-phenyl)propane-1,3-dione | 1-(4-fluorophenyl)-3-(2-hydroxy-5-methoxyphenyl)propane-1,3-dione | 1-(4-fluorophenyl)-3-(5-methoxy-2-oxidanyl-phenyl)propane-1,3-dione | MLS000108321 | SMR000104281 | cid_768764
Type:
Small organic molecule
Emp. Form.:
C16H13FO4
Mol. Mass.:
288.2704
SMILES:
COc1ccc(O)c(c1)C(=O)CC(=O)c1ccc(F)cc1
Structure:
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