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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48214
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
3930±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48214
Synonyms:
3-(5-Ethyl-benzooxazol-2-yl)-phenylamine | 3-(5-ethyl-1,3-benzoxazol-2-yl)aniline | MLS000525240 | SMR000122114 | [3-(5-ethyl-1,3-benzoxazol-2-yl)phenyl]amine | cid_735963
Type:
Small organic molecule
Emp. Form.:
C15H14N2O
Mol. Mass.:
238.2845
SMILES:
CCc1ccc2oc(nc2c1)-c1cccc(N)c1
Structure:
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