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Target
D(1A) dopamine receptor
Ligand
BDBM49079
Substrate
n/a
Meas. Tech.
Allosteric Modulators of D1 Receptors: Dose-dependent Assay
EC50
0.00428±n/a nM
Citation
 PubChem, PC Allosteric Modulators of D1 Receptors: Dose-dependent Assay PubChem Bioassay (2007)[AID] 
Target
Name:
D(1A) dopamine receptor
Synonyms:
DA D1 receptor | DOPAMINE D1 | DRD1 | DRD1_HUMAN | Dopamine D1 receptor | Dopamine D1 receptor (D1R) | Dopamine D1A
Type:
Enzyme
Mol. Mass.:
49303.43
Organism:
Homo sapiens (Human)
Description:
P21728
Residue:
446
Sequence:
MRTLNTSAMDGTGLVVERDFSVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPTSPSDGNATSLAETIDNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNCQTTTGNGKPVECSQPESSFKMSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCGSGETQPFCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPATNNAIETVSINNNGAAMFSSHHEPRGSISKECNLVYLIPHAVGSSEDLKKEEAAGIARPLEKLSPALSVILDYDTDVSLEKIQPITQNGQHPT
  
Inhibitor
Name:
BDBM49079
Synonyms:
3-amino-5-phenyl-2-thiophenecarboxylic acid ethyl ester | 3-amino-5-phenyl-thiophene-2-carboxylic acid ethyl ester | MLS000058832 | SMR000069098 | cid_838333 | ethyl 3-amino-5-phenyl-2-thiophenecarboxylate | ethyl 3-amino-5-phenylthiophene-2-carboxylate | ethyl 3-azanyl-5-phenyl-thiophene-2-carboxylate
Type:
Small organic molecule
Emp. Form.:
C13H13NO2S
Mol. Mass.:
247.313
SMILES:
CCOC(=O)c1sc(cc1N)-c1ccccc1
Structure:
Search PDB for entries with ligand similarity: