Reaction Details Report a problem with these data
Target
POsterior Segregation
Ligand
BDBM52919
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM52919
Synonyms:
2-(5,7-Dinitro-quinolin-8-ylamino)-benzoic acid | 2-[(5,7-dinitro-8-quinolinyl)amino]benzoic acid | 2-[(5,7-dinitro-8-quinolyl)amino]benzoic acid | 2-[(5,7-dinitroquinolin-8-yl)amino]benzoic acid | MLS000806875 | SMR000414684 | cid_3763920
Type:
Small organic molecule
Emp. Form.:
C16H10N4O6
Mol. Mass.:
354.2738
SMILES:
OC(=O)c1ccccc1Nc1c(cc([N+]([O-])=O)c2cccnc12)[N+]([O-])=O
Structure:
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