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Target
POsterior Segregation
Ligand
BDBM53059
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA
EC50
24385±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of POS-1 Binding to mex-3-RNA PubChem Bioassay (2009)[AID] 
Target
Name:
POsterior Segregation
Synonyms:
POsterior Segregation family member (pos-1)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
29838.90
Organism:
Caenorhabditis elegans
Description:
gi_17562800
Residue:
264
Sequence:
MADNDFLSGEAIMVFKKEILDSHSDFTRSLSHQSASPEAYDQENVFSQDFQPFMKQDKETQNSASQPTSEQSLANRDPCTVPDDLREEMMRQRRKEDAFKTALCDAYKRSQACSYGDQCRFAHGVHELRLPMNPRGRNHPKYKTVLCDKFSMTGNCKYGTRCQFIHKIVDGNAAKLASGAHANTSSKSPARNAAAHNHSLFVPQGSTDRSMDLNQSLPIRQSDLVRAFARATRLDVSGYNSTAQLAQYFESQFQRIQQLSSHHH
  
Inhibitor
Name:
BDBM53059
Synonyms:
2-(7-Nitro-benzo[1,2,5]oxadiazol-4-ylamino)-phenol | 6-[(4-nitro-1,3-dihydro-2,1,3-benzoxadiazol-7-yl)imino]-1-cyclohexa-2,4-dienone | 6-[(4-nitro-1,3-dihydro-2,1,3-benzoxadiazol-7-yl)imino]cyclohexa-2,4-dien-1-one | 6-[(7-nitro-1,3-dihydrobenzofurazan-4-yl)imino]cyclohexa-2,4-dien-1-one | MLS001206694 | SMR000516446 | cid_5719582
Type:
Small organic molecule
Emp. Form.:
C12H8N4O4
Mol. Mass.:
272.2163
SMILES:
[O-]c1ccccc1\N=c1/ccc([N+]([O-])=O)c2[nH]o[nH+]c12
Structure:
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